SCHEMBL19586554

SCHEMBL19586554

O=C(O)N1CCC2(CCCN2Cc2ccccc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.49
MGLL Q99685 2/20 0.47
CYP2D6 P10635 5/20 0.47
ALDH1A1 P00352 4/20 0.45
CYP3A4 P08684 3/20 0.45
USP2 O75604 1/20 0.45
CHRM2 P08172 2/20 0.45
CHRM3 P20309 1/20 0.45
TSHR P16473 1/20 0.43
FAAH O00519 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1556555 0.92 EPHX2 (0.53) EPHX2MGLLCYP2D6ALDH1A1CYP3A4
SCHEMBL19603318 0.87 MGLL (0.48) MGLLFAAH
SCHEMBL23968905 0.85 OPRD1 (0.51) EPHX2MGLLCYP2D6ALDH1A1
SCHEMBL23642541 0.85 OPRD1 (0.51) EPHX2MGLLCYP2D6ALDH1A1CYP3A4
SCHEMBL18711496 0.83 CYP2D6 (0.58) EPHX2CYP2D6ALDH1A1CYP3A4USP2
SCHEMBL14891885 0.82 EPHX2 (0.64) EPHX2CYP2D6ALDH1A1CYP3A4USP2
SCHEMBL18702131 0.80 EPHX2 (0.48) EPHX2MGLLCYP2D6ALDH1A1CYP3A4
SCHEMBL19582609 0.79 MGLL (0.74) MGLL
SCHEMBL30924710 0.79 SIGMAR1 (0.45) EPHX2ALDH1A1CYP3A4TSHR
SCHEMBL1557924 0.79 KMT2A (0.49) EPHX2CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3455226-B1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME LUNDBECK LA JOLLA RESEARCH CENTER INC (US) 2020-12-30 EP disclosed
EP-3455226-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME Abide Therapeutics, Inc. (US) 2019-03-20 EP disclosed
WO-2017197192-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2017-11-16 WO disclosed