SCHEMBL19590653

SCHEMBL19590653

CCc1cc(C(=O)NC(C)(C)C)cc(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
GAA P10253 1/20 0.41
CES2 O00748 1/20 0.41
ANO1 Q5XXA6 2/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
DDR1 Q08345 3/20 0.40
MLYCD O95822 1/20 0.40
TACR1 P25103 1/20 0.40
CACNA1H O95180 1/20 0.39
TP53BP1 Q12888 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21028343 0.88 LMNA (0.42) ALDH1A1LMNAHTTCACNA1H
SCHEMBL20877084 0.85 CES2 (0.55) NOTUMGAACES2ANO1DDR1
SCHEMBL17789598 0.85 MEN1 (0.44) POLBLMNAHTTCACNA1H
SCHEMBL19590713 0.82 KMT2A (0.39) ANO1LMNAHTTCACNA1H
SCHEMBL16142872 0.81 NOTUM (0.62) NOTUMGAACES2ANO1ALDH1A1
SCHEMBL13753158 0.80 DDR1 (0.47) NOTUMGAACES2ANO1POLB
SCHEMBL15726944 0.80 ADCY8 (0.46) NOTUMGAACES2ANO1HTT
SCHEMBL19590866 0.79 TP53 (0.43) LMNADDR1CACNA1H
SCHEMBL21697648 0.79 RXRA (0.52) NOTUMCES2ALDH1A1POLBMLYCD
SCHEMBL17897037 0.79 MRGPRX4 (0.51) NOTUMCES2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9815851-B2 Pyrrolo carboxamides as modulators of orphan nuclear receptor RAR-related orphan receptor-gamma (RORγ, NR1F3) activity and for the treatment of chronic inflammatory and autoimmune diseases PHENEX PHARMACEUTICALS AG (DE) 2017-11-14 US disclosed