SCHEMBL19620983

SCHEMBL19620983

CCCC(/C=C(/C)NC=O)=C(/C)CNC(=O)c1cc(OCCN2CCOCC2)cc2c1ccn2C(C)C

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.35
GAA P10253 1/20 0.35
ACACB O00763 1/20 0.35
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 3/20 0.35
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
THRB P10828 5/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
THRA P10827 1/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
MET P08581 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14717434 0.76 KDM4E (0.48) SMN1; SMN2GAAACACBALDH1A1KDM4E
SCHEMBL14727056 0.73 EZH2 (0.58)
SCHEMBL19620960 0.69 EZH2 (0.33)
SCHEMBL19620781 0.69 LMNA (0.32) LMNA
SCHEMBL14717102 0.68 KDM4E (0.47) GAAALDH1A1KDM4EKMT2A
SCHEMBL14717869 0.67 PRKAB2 (0.46) SMN1; SMN2GAAALDH1A1KDM4EMAPT
SCHEMBL17956112 0.63 EZH2 (0.52)
SCHEMBL21666232 0.61 SMN1; SMN2 (0.53) SMN1; SMN2GAAALDH1A1KDM4ENPC1
SCHEMBL863522 0.59 SMN1; SMN2 (0.81) SMN1; SMN2GAAALDH1A1KDM4ETHRB
SCHEMBL11204217 0.59 THRB (0.79) SMN1; SMN2GAAALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246027-A1 INDOLE DERIVATIVES FOR THE TREATMENT OF CANCER GlaxoSmithKline LLC (US) 2017-11-22 EP disclosed