SCHEMBL19623723

SCHEMBL19623723

CN(CCCN1CCCOCC1)c1ccc(N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.43
NPSR1 Q6W5P4 1/20 0.40
HTR7 P34969 6/20 0.39
HRH3 Q9Y5N1 4/20 0.39
MAPK1 P28482 2/20 0.39
CHRM1 P11229 2/20 0.39
HTR2A P28223 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CHRM2 P08172 1/20 0.39
SCN1A P35498 1/20 0.39
HTR2B P41595 1/20 0.39
KCNH2 Q12809 1/20 0.39
SCN2A Q99250 1/20 0.39
SCN3A Q9NY46 1/20 0.39
POLB P06746 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
KEAP1 Q14145 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
USP2 O75604 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2375987 0.95 HTR7 (0.42) SIGMAR1NPSR1HTR7HRH3MAPK1
SCHEMBL2375260 0.86 SIGMAR1 (0.46) SIGMAR1HTR7HRH3MAPK1CHRM1
SCHEMBL2377649 0.80 LMNA (0.50) SIGMAR1HTR7ALDH1A1LMNA
SCHEMBL3576244 0.78 SIGMAR1 (0.60) SIGMAR1HRH3CHRM1HTR2AALDH1A1
SCHEMBL3225925 0.78 KDM4E (0.46) NPSR1HRH3MAPK1ALDH1A1SMN1; SMN2
SCHEMBL3562916 0.77 SIGMAR1 (0.59) SIGMAR1HRH3CHRM1HTR2AALDH1A1
SCHEMBL2376367 0.75 MAPT (0.58) SIGMAR1HTR7ALDH1A1CYP1A2POLB
SCHEMBL13103802 0.73 POLB (0.48) ALDH1A1POLBSMN1; SMN2
SCHEMBL2157801 0.72 ALDH1A1 (0.51) SIGMAR1HRH3MAPK1CHRM1HTR2A
SCHEMBL11440371 0.71 HTR7 (0.53) SIGMAR1HTR7ALDH1A1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed