SCHEMBL19624951

SCHEMBL19624951

[N-]=[N+]=NCc1ccc2cc(C(=O)N=N)[nH]c2c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 1/20 0.36
IDO1 P14902 2/20 0.35
PLG P00747 1/20 0.34
PLAU P00749 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
ALOX15 P16050 4/20 0.33
FLT3 P36888 2/20 0.33
EIF4A3 P38919 1/20 0.33
DAO P14920 1/20 0.33
RHEB Q15382 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19625002 0.80 MCL1 (0.35)
SCHEMBL19624948 0.74 HTR6 (0.39) IDO1FLT3DAOKDM4EALDH1A1
SCHEMBL23458852 0.73 CYP2A6 (0.45) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL29965121 0.73 CYP2A6 (0.45) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL19624933 0.72 HRH4 (0.51) FLT3
SCHEMBL12786510 0.70 HRH4 (0.55) ALOX15ALDH1A1
SCHEMBL31440929 0.67 AHR (0.42) KDM4EALDH1A1MAPK1
SCHEMBL19625088 0.67 MCL1 (0.33)
SCHEMBL30489877 0.65 HDAC3 (0.35) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL31440882 0.64 AHR (0.42) HDAC1HDAC8ALOX15GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2892880-B1 INDOLE CARBOXAMIDE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2017-11-22 EP disclosed