SCHEMBL19632072

SCHEMBL19632072

CC(=O)NSc1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.44
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
NR4A1 P22736 1/20 0.42
NR4A2 P43354 1/20 0.42
NR4A3 Q92570 1/20 0.42
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
IDO1 P14902 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
SRD5A2 P31213 1/20 0.39
DHODH Q02127 1/20 0.39
KIF11 P52732 1/20 0.39
HDAC3 O15379 1/20 0.39
ADAM17 P78536 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27651930 0.81 KIF11 (0.50) EPHX2CES2CES1ALDH1A1IDO1
SCHEMBL7536726 0.76 HPGD (0.35) ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL7536730 0.76 ALDH1A1 (0.48) ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL19311702 0.76 TDP1 (0.48) CES2CES1ALDH1A1LMNAADORA3
SCHEMBL24713130 0.75 EPHX2 (0.58) EPHX2LMNAHTTTRPV1
SCHEMBL28037693 0.75 TEAD1 (0.43) CES2CES1ALDH1A1LMNAHTT
SCHEMBL10431593 0.74 MTNR1A (0.48) CES2CES1ALDH1A1LMNASMN1; SMN2
SCHEMBL26679563 0.73 KIF11 (0.46) EPHX2CES2CES1ALDH1A1KIF11
SCHEMBL669442 0.71 EPHX2 (0.70) EPHX2ALDH1A1LMNAHTTIDO1
Hydrochloric Acid SCHEMBL28845768 0.71 MTNR1A (0.47) ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017201155-A1 lSOXAZOLE DERIVATIVES AS FXR AGONISTS AND METHODS OF USE THEREOF ENANTA PHARMACEUTICALS, INC. (US) 2017-11-23 WO disclosed