SCHEMBL19633656

SCHEMBL19633656

COc1ccc2c(Nc3cccc([N+](=O)[O-])c3)ccnc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.58
AKR1C2 P52895 1/20 0.58
GAK O14976 2/20 0.57
RIPK2 O43353 1/20 0.57
COQ8A Q8NI60 1/20 0.57
NLK Q9UBE8 1/20 0.57
ABCG2 Q9UNQ0 5/20 0.53
PTK6 Q13882 3/20 0.53
PDGFRA P16234 1/20 0.52
KDR P35968 1/20 0.52
HTR1A P08908 2/20 0.51
ADRA1D P25100 2/20 0.51
ADRA1A P35348 2/20 0.51
ADRA1B P35368 2/20 0.51
MITF O75030 1/20 0.51
LMNA P02545 1/20 0.51
KMT2A Q03164 1/20 0.51
ERBB2 P04626 3/20 0.49
GSK3A P49840 1/20 0.49
GSK3B P49841 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633573 0.90 KMT2A (0.49) AKR1C3AKR1C2GAKRIPK2COQ8A
SCHEMBL19633684 0.89 KMT2A (0.64) AKR1C3AKR1C2GAKRIPK2COQ8A
SCHEMBL19633806 0.88 KMT2A (0.51) AKR1C3AKR1C2GAKRIPK2COQ8A
SCHEMBL19633549 0.87 KMT2A (0.55) AKR1C3AKR1C2GAKRIPK2COQ8A
SCHEMBL19633777 0.86 GAK (0.57) AKR1C3AKR1C2GAKRIPK2COQ8A
SCHEMBL19633569 0.85 KMT2A (0.52) AKR1C3AKR1C2ABCG2PTK6PDGFRA
SCHEMBL19633676 0.84 GAK (0.68) GAKRIPK2COQ8ANLKABCG2
SCHEMBL9069952 0.84 GAK (0.63) AKR1C3AKR1C2GAKRIPK2COQ8A
SCHEMBL19633574 0.84 CTSV (0.56) ABCG2PTK6MITFLMNAKMT2A
SCHEMBL19633621 0.84 KMT2A (0.49) AKR1C3AKR1C2ABCG2PTK6PDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed