SCHEMBL19633690

SCHEMBL19633690

FC(F)(F)c1cc(Nc2ccnc3cc(OCCCc4ccccc4)ccc23)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 4/20 0.47
CCNC P24863 1/20 0.46
CDK8 P49336 1/20 0.46
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
RIPK2 O43353 2/20 0.43
COQ8A Q8NI60 2/20 0.43
NLK Q9UBE8 2/20 0.43
ALK Q9UM73 4/20 0.42
ERBB2 P04626 1/20 0.41
HRH3 Q9Y5N1 2/20 0.40
DNMT1 P26358 1/20 0.40
DNMT3A Q9Y6K1 1/20 0.40
EPHB6 O15197 1/20 0.40
ABL1 P00519 1/20 0.40
LCK P06239 1/20 0.40
EPHA1 P21709 1/20 0.40
EPHA8 P29322 1/20 0.40
TXK P42681 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633682 0.92 GSK3A (0.52) GAKCCNCCDK8GSK3AGSK3B
SCHEMBL19633681 0.92 CCNC (0.51) GAKCCNCCDK8GSK3AGSK3B
SCHEMBL19633566 0.82 SIRT2 (0.47) GAKALKERBB2SIRT2KDR
SCHEMBL19633687 0.82 ERBB2 (0.49) GAKRIPK2COQ8ANLKALK
SCHEMBL19633503 0.80 GAK (0.53) GAKGSK3AGSK3BRIPK2COQ8A
SCHEMBL19633692 0.78 CCNC (0.50) CCNCCDK8ALKERBB2HRH3
SCHEMBL19633545 0.77 KMT2A (0.49) CCNCCDK8ALKERBB2KDM4E
SCHEMBL19633778 0.76 GAK (0.69) GAKGSK3AGSK3BRIPK2COQ8A
SCHEMBL27969044 0.73 MAOA (0.50) KDM4EMEN1ALDH1A1LMNAGLA
SCHEMBL29200458 0.72 GAK (0.64) GAKCCNCCDK8GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed