SCHEMBL19634004

SCHEMBL19634004

OCc1cc(C(F)F)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.36
GCGR P47871 1/20 0.36
KIF11 P52732 1/20 0.35
MAPK1 P28482 1/20 0.35
MAP2K4 P45985 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
MAPKAPK3 Q16644 1/20 0.35
MAPK6 Q16659 1/20 0.35
DPP4 P27487 1/20 0.34
ADRB2 P07550 6/20 0.33
S1PR1 P21453 1/20 0.33
ADRB1 P08588 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
HIF1A Q16665 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRB3 P13945 1/20 0.33
ADRA2B P18089 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11994355 0.86 GCGR (0.41) GCGRKIF11MAPK1MAP2K4MAPKAPK2
SCHEMBL18914333 0.83 MRGPRX4 (0.36) MRGPRX4KIF11S1PR1CYP1A2TSHR
SCHEMBL29738108 0.83 MRGPRX4 (0.36) MRGPRX4KIF11S1PR1CYP1A2TSHR
SCHEMBL16638758 0.81 DPP4 (0.39) MRGPRX4KIF11DPP4ADRB1CYP2D6
SCHEMBL19568082 0.79 DPP4 (0.34) MRGPRX4KIF11DPP4
SCHEMBL13185576 0.79 TRPV4 (0.35) MRGPRX4DPP4S1PR1ADRB1ADRA2A
SCHEMBL20256735 0.79 DPP4 (0.38) MRGPRX4KIF11DPP4CYP2D6
SCHEMBL13160946 0.78 GABRA1 (0.41) DPP4CYP2D6
SCHEMBL6499247 0.77 MAPK1 (0.35) GCGRMAPK1MAP2K4MAPKAPK2MAPKAPK3
SCHEMBL19566851 0.76 HRH4 (0.33) GCGRDPP4ADRB1ADRA2AADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017201468-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-11-23 WO disclosed