SCHEMBL19634692

SCHEMBL19634692

CC(=O)NCc1ccc(C(=O)N(CCN(C)C)CCN(C)C)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.57
HDAC1 Q13547 10/20 0.54
HDAC6 Q9UBN7 5/20 0.54
ALDH1A1 P00352 3/20 0.53
POLB P06746 1/20 0.53
MAPT P10636 1/20 0.53
RAB9A P51151 1/20 0.53
HDAC3 O15379 6/20 0.47
HDAC2 Q92769 6/20 0.47
EPHX2 P34913 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
LIMK2 P53671 1/20 0.44
HDAC8 Q9BY41 5/20 0.44
HDAC4 P56524 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HTR5A P47898 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634448 0.86 KMT2A (0.58) KMT2AHDAC1HDAC6ALDH1A1POLB
SCHEMBL23471131 0.86 KMT2A (0.62) KMT2AHDAC1HDAC6ALDH1A1POLB
SCHEMBL19634696 0.85 KMT2A (0.54) KMT2AHDAC1HDAC6ALDH1A1POLB
SCHEMBL23471262 0.84 KMT2A (0.55) KMT2AHDAC1HDAC6ALDH1A1POLB
SCHEMBL19634729 0.83 HDAC3 (0.47) KMT2AHDAC1HDAC6RAB9AHDAC3
SCHEMBL23471106 0.82 HDAC1 (0.55) KMT2AHDAC1HDAC6ALDH1A1POLB
SCHEMBL19682898 0.82 KMT2A (0.66) KMT2AHDAC1HDAC6ALDH1A1POLB
SCHEMBL21015203 0.82 EPHX2 (0.41) KMT2AHDAC1HDAC6ALDH1A1RAB9A
SCHEMBL19634445 0.80 ALDH1A1 (0.51) KMT2AHDAC1HDAC6ALDH1A1POLB
SCHEMBL23470991 0.79 HDAC1 (0.62) KMT2AHDAC1HDAC6ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed