SCHEMBL19639792

SCHEMBL19639792

Cn1c(-c2ncnn2-c2ccc(C#N)cc2)c(C(=O)O)c(=O)n1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 15/20 0.46
CYP2C9 P11712 5/20 0.41
CTSK P43235 4/20 0.41
CYP3A4 P08684 3/20 0.41
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19639807 0.90 ELANE (0.48) ELANECYP2C9CYP3A4
SCHEMBL19639806 0.86 ELANE (0.43) ELANECYP2C9CTSKCYP3A4
SCHEMBL19639818 0.86 ELANE (0.44) ELANECYP2C9CYP3A4
SCHEMBL19639985 0.85 ELANE (0.56) ELANECYP2C9CTSKCYP3A4POLB
SCHEMBL19639793 0.79 PFKFB3 (0.33) ELANE
SCHEMBL17819296 0.79 ELANE (0.50) ELANECYP2C9CTSKCYP3A4POLB
SCHEMBL19684694 0.79 ELANE (0.56) ELANECYP2C9CTSKCYP3A4
SCHEMBL19688568 0.78 ELANE (0.41) ELANECYP2C9CYP3A4
SCHEMBL21796123 0.77 ELANE (0.54) ELANECYP2C9CTSKCYP3A4
SCHEMBL19640024 0.77 ELANE (0.54) ELANECYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464269-B1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF A HNE RELATED DISEASE CHIESI FARM SPA (IT) 2020-04-01 EP disclosed
WO-2017207433-A9 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF A DISEASE IN WHICH HNE IS IMPLICATED CHIESI FARMACEUTICI S.P.A. (IT) 2018-03-01 WO disclosed
US-9862706-B2 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2018-01-09 US disclosed
US-9862706-B2 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2018-01-09 US disclosed
WO-2017207433-A1 HETETOCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF A DISEASE IN WHICH HNE IS IMPLICATED CHIESI FARMACEUTICI S.P.A. (IT) 2017-12-07 WO disclosed
US-20170342056-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2017-11-30 US disclosed
US-20170342056-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2017-11-30 US disclosed
US-20170342056-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2017-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170342056-A1 NOVEL COMPOUNDS SERPINB1, ELANE, MPO ELANE 2/4885CYP2C9 2925/4885CTSK 100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.