SCHEMBL1966198

SCHEMBL1966198

O=Cc1nocc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.44
HSP90AA1 P07900 1/20 0.42
GSR P00390 1/20 0.38
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
NPC1 O15118 3/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 2/20 0.35
RAB9A P51151 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GPR55 Q9Y2T6 2/20 0.34
NTSR1 P30989 1/20 0.34
PTPN1 P18031 3/20 0.34
PTPN2 P17706 2/20 0.34
IP6K1 Q92551 1/20 0.33
NOTUM Q6P988 1/20 0.33
CYP2A6 P11509 1/20 0.33
TDO2 P48775 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15873926 0.81 KDM4E (0.42) PTGS2NPC1ALDH1A1POLBRAB9A
SCHEMBL27752586 0.75 TDO2 (0.39) ALDH1A1CYP2A6TDO2
SCHEMBL27773472 0.73 ALDH1A1 (0.38) MEN1KMT2ANPC1ALDH1A1POLB
SCHEMBL27773454 0.72 DPP4 (0.40) MEN1KMT2ANPC1ALDH1A1RAB9A
SCHEMBL1797330 0.71 PTGS2 (0.67) PTGS2HSP90AA1MEN1KMT2AGPR55
SCHEMBL6630764 0.69 HSP90AA1 (0.46) PTGS2HSP90AA1NPC1ALDH1A1RAB9A
SCHEMBL6630766 0.69 PTGS2 (0.47) PTGS2HSP90AA1MEN1KMT2ANPC1
SCHEMBL2797055 0.69 LMNA (0.59) PTGS2HSP90AA1NPC1ALDH1A1RAB9A
SCHEMBL2886350 0.69 HSP90AA1 (0.54) PTGS2HSP90AA1MEN1KMT2ANPC1
SCHEMBL5729643 0.69 HSP90AA1 (0.46) PTGS2HSP90AA1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334636-A2 HYDROXAMIC ACID DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS Pfizer Inc. (US) 2011-06-22 EP disclosed
WO-2010032147-A2 HYDROXAMIC ACID DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS PFIZER INC. (US) 2010-03-25 WO disclosed
CN-1135210-C Process for preparation of 1-aryl-3-cyclopropyl-1,3-propanediones ����-���ʿ�ũҵ��˾ 2004-01-21 CN disclosed
CN-1262670-A Preparation method of 1-aryl-3-cyclopropyl-1, 3-propanedione RHONE POULENC AGROCHIMIE (FR) 2000-08-09 CN disclosed