SCHEMBL19664705

SCHEMBL19664705

O=C(O)C(Cc1ccccc1)c1ccncn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPA1 P15085 6/20 0.49
CYP1A2 P05177 1/20 0.49
P4HTM Q9NXG6 1/20 0.48
CPA3 P15088 3/20 0.44
CPB2 Q96IY4 2/20 0.44
FOLH1 Q04609 1/20 0.44
CPB1 P15086 1/20 0.44
EPHX1 P07099 1/20 0.42
ALPI P09923 1/20 0.42
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.42
XIAP P98170 1/20 0.42
SLC7A5 Q01650 1/20 0.42
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127361 0.82 CYP1A2 (0.53) CPA1CYP1A2P4HTMCPA3CPB2
SCHEMBL1888804 0.79 CPA1 (0.53) CPA1CYP1A2P4HTMCPA3CPB2
SCHEMBL28092231 0.79 L3MBTL1 (0.41) CPA1CYP1A2CPA3CPB2CPB1
SCHEMBL17825462 0.75 P4HTM (0.54) CPA1CYP1A2P4HTMCPA3CPB2
SCHEMBL17479494 0.74 P4HTM (0.50) CPA1CYP1A2P4HTMCPA3CPB2
SCHEMBL7816162 0.73 CHRM1 (0.61) CPA1CYP1A2P4HTMEPHX1SLC6A2
SCHEMBL7816160 0.73 CHRM1 (0.61) CPA1CYP1A2P4HTMEPHX1SLC6A2
SCHEMBL7346172 0.73 CYP1A2 (0.77) CPA1CYP1A2CPA3CPB2FOLH1
SCHEMBL11643934 0.73 P2RX7 (0.38) CYP1A2PKMALDH1A1CYP3A4
SCHEMBL1127590 0.73 KMT2A (0.46) CYP1A2P4HTMSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091940-B3 4-PHENYL-6-(2,2,2-TRIFLUORO-1-PHENYLETHOXY)PYRIMIDINE-BASED COMPOUNDS AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS INC (US) 2017-12-06 EP disclosed