SCHEMBL19675178

SCHEMBL19675178

CS(=O)(=O)OCc1ccc2c(c1)CNC2

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
HTR6 P50406 2/20 0.41
PNMT P11086 6/20 0.40
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
CA1 P00915 1/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
USP28 Q96RU2 1/20 0.32
MLNR O43193 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16648351 0.78 DRD2 (0.37) DRD2DRD3HTR6CA2
SCHEMBL27538780 0.77 DRD2 (0.38) DRD2DRD3CA2CA9CA1
Hydrochloric Acid SCHEMBL4715513 0.76 DRD2 (0.36) DRD2DRD3HTR6CA2
SCHEMBL20323430 0.76 DAPK3 (0.42) CA9
SCHEMBL29868930 0.74 KMT2A (0.45) DRD2DRD3HTR6PNMTHTR2A
SCHEMBL4952656 0.74 CA2 (0.58) CA2CA9CA1
Hydrochloric Acid SCHEMBL29868424 0.74 DRD2 (0.41) DRD2DRD3HTR6PNMTHTR2A
SCHEMBL20672086 0.73 DRD2 (0.35) DRD2DRD3HTR6MLNR
SCHEMBL28277152 0.73 DRD2 (0.35) DRD2DRD3HTR6PNMT
Hydrochloric Acid SCHEMBL4716276 0.73 DRD2 (0.37) DRD2DRD3HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3252050-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed
EP-3252049-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed