SCHEMBL28277152

SCHEMBL28277152

O=COCc1ccc2c(c1)CNC2

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
HTR6 P50406 1/20 0.35
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
ITGB3 P05106 2/20 0.31
ITGA2B P08514 2/20 0.31
PLAU P00749 1/20 0.31
TYK2 P29597 1/20 0.31
PNMT P11086 1/20 0.31
RXRB P28702 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28255640 0.79 HTT (0.38) TYK2PNMT
SCHEMBL27645613 0.77 RXRB (0.50) RXRB
SCHEMBL16648351 0.77 DRD2 (0.37) DRD2DRD3HTR6PLAU
Hydrochloric Acid SCHEMBL4715513 0.75 DRD2 (0.36) DRD2DRD3HTR6ITGB3ITGA2B
SCHEMBL28869247 0.74 NTRK2 (0.45) DRD2TYK2
SCHEMBL19675178 0.73 DRD2 (0.41) DRD2DRD3HTR6PNMT
Hydrochloric Acid SCHEMBL4716276 0.72 DRD2 (0.37) DRD2DRD3HTR6ITGB3ITGA2B
SCHEMBL20672086 0.72 DRD2 (0.35) DRD2DRD3HTR6PLAU
SCHEMBL28835938 0.72 SMN1; SMN2 (0.40) DRD2
SCHEMBL28071113 0.72 DRD2 (0.49) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104045552-B Medicinal compound as neuroprotective agent 江苏先声药业有限公司 2019-06-11 CN disclosed
CN-109265443-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-01-25 CN disclosed