SCHEMBL19675765

SCHEMBL19675765

Cc1cc(N)ccc1C1NNC(=O)c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PBRM1 Q86U86 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
PTPRC P08575 2/20 0.37
HPGD P15428 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
APAF1 O14727 1/20 0.37
TDP2 O95551 1/20 0.37
NSD2 O96028 1/20 0.37
LMNA P02545 1/20 0.37
PLA2G1B P04054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19675735 0.79 HSD17B10 (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL19675259 0.76 PARP3 (0.39) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL19675283 0.73 BRD4 (0.36) PBRM1TNKS2KMT2AMEN1CYP1A2
SCHEMBL29016841 0.69 PBRM1 (0.60) ALDH1A1NPC1TSHRPBRM1TNKS2
SCHEMBL10438247 0.67 NPC1 (0.40) ALDH1A1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL19675124 0.65 S100A4 (0.40) ALDH1A1SMN1; SMN2TSHRPBRM1TNKS2
SCHEMBL4802137 0.65 HTR2A (0.39) ALDH1A1SMN1; SMN2TSHRPBRM1TNKS2
SCHEMBL19675594 0.65 CYP26A1 (0.39) ALDH1A1CYP3A4PBRM1KMT2AMEN1
SCHEMBL1335484 0.65 KDR (0.59) PARP1
Phthalimide SCHEMBL27407474 0.65 PDE10A (0.61) ALDH1A1NPC1RAB9ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3252050-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed
EP-3252049-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed