SCHEMBL19682384

SCHEMBL19682384

O=C1CCCc2c(Cl)ccc(S(=O)(=O)Cl)c21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
RRM1 P23921 1/20 0.38
RRM2B Q7LG56 1/20 0.38
BRD4 O60885 7/20 0.38
DYRK1A Q13627 1/20 0.35
BRDT Q58F21 2/20 0.35
BRD9 Q9H8M2 2/20 0.35
BRD7 Q9NPI1 2/20 0.35
CREBBP Q92793 1/20 0.35
CECR2 Q9BXF3 1/20 0.35
ALDH1A1 P00352 3/20 0.33
TRPV4 Q9HBA0 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 2/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
POLB P06746 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24542960 0.74 BRD4 (0.42) CHRM2CHRM1RRM1RRM2BBRD4
SCHEMBL9040886 0.74 BRD4 (0.43) BRD4DYRK1ABRDTBRD9BRD7
SCHEMBL19682389 0.74 BRD4 (0.40) BRD4DYRK1ABRDTBRD9BRD7
SCHEMBL16555610 0.71 EPAS1 (0.42) ALDH1A1TRPV4KDM4EGAATSHR
SCHEMBL19682938 0.71 CHRM2 (0.40) CHRM2CHRM1RRM1RRM2BALDH1A1
SCHEMBL7659144 0.69 MAPT (0.46) BRD4ALDH1A1SMN1; SMN2LMNAPOLB
SCHEMBL7103532 0.67 BRD4 (0.43) BRD4DYRK1ABRDTBRD9BRD7
SCHEMBL31104321 0.67 BRD4 (0.40) BRD4DYRK1ABRDTBRD9BRD7
SCHEMBL2370165 0.67 KDM4E (0.45) BRD4DYRK1ABRDTBRD9BRD7
SCHEMBL6686475 0.67 BRD4 (0.42) CHRM2CHRM1RRM1RRM2BBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 CHRM2 4302/4885CHRM1 4399/4885RRM1 5/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 CHRM2 4302/4885CHRM1 4399/4885RRM1 5/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 CHRM2 4302/4885CHRM1 4399/4885RRM1 5/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B CHRM2 4208/4885CHRM1 4101/4885RRM1 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.