SCHEMBL19682597

SCHEMBL19682597

Cc1c(F)cccc1[C@@H](C)[C@H](N)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPP7 Q9UHL4 3/20 0.40
DPP4 P27487 1/20 0.40
SLC1A1 P43005 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
GAA P10253 1/20 0.36
SLC7A5 Q01650 1/20 0.35
LMNA P02545 1/20 0.35
HIF1A Q16665 1/20 0.35
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
DPP8 Q6V1X1 2/20 0.34
DPP9 Q86TI2 2/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20889385 1.00 DPP7 (0.40) DPP7DPP4SLC1A1SMN1; SMN2GAA
SCHEMBL19682604 0.85 CES2 (0.45) DPP7DPP4SLC1A1SMN1; SMN2GAA
SCHEMBL20889267 0.85 CES2 (0.45) DPP7DPP4SLC1A1SMN1; SMN2GAA
SCHEMBL20889256 0.85 GRM1 (0.37) DPP7DPP4SLC1A1SLC7A5AKR1C3
SCHEMBL19682749 0.85 GRM1 (0.37) DPP7DPP4SLC1A1SLC7A5AKR1C3
SCHEMBL19682745 0.83 SLC1A3 (0.40) SLC1A1SLC7A5LMNA
SCHEMBL20889380 0.83 SLC1A3 (0.40) SLC1A1SLC7A5LMNA
SCHEMBL20889384 0.83 DPP4 (0.39) DPP7DPP4SLC1A1SMN1; SMN2GAA
SCHEMBL19682586 0.83 DPP4 (0.39) DPP7DPP4SLC1A1SMN1; SMN2GAA
SCHEMBL503246 0.81 GRM1 (0.50) SMN1; SMN2GAACES2CES1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
EP-3466934-A1 SULFONAMIDE COMPOUND OR SALT THEREOF Taiho Pharmaceutical Co., Ltd. (JP) 2019-04-10 EP disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 DPP7 3961/4885DPP4 3280/4885SLC1A1 3403/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 DPP7 3961/4885DPP4 3280/4885SLC1A1 3403/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 DPP7 3961/4885DPP4 3280/4885SLC1A1 3403/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B DPP7 4703/4885DPP4 4367/4885SLC1A1 3066/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.