SCHEMBL19682602

SCHEMBL19682602

C[C@H](c1cccc2sccc12)[C@H](N)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.42
SLC1A3 P43003 4/20 0.35
SLC1A2 P43004 4/20 0.35
SLC1A1 P43005 4/20 0.35
APP P05067 1/20 0.34
SLC9A1 P19634 1/20 0.34
SYK P43405 1/20 0.34
GPR139 Q6DWJ6 3/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
CSNK2A1 P68400 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
SLC7A5 Q01650 1/20 0.32
CYP2C9 P11712 3/20 0.32
LMNA P02545 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
PTGS1 P23219 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20889266 1.00 ALOX5 (0.42) ALOX5SLC1A3SLC1A2SLC1A1APP
SCHEMBL10367027 0.83 CXCL8 (0.41) ALOX5APPGPR139CSNK2A2CSNK2B
SCHEMBL10928021 0.81 ALOX5 (0.36) ALOX5APPSYKCSNK2A2CSNK2B
SCHEMBL14622826 0.81 ALOX5 (0.59) ALOX5SLC1A3SLC1A2SLC1A1APP
SCHEMBL19682606 0.81 ALOX5 (0.59) ALOX5SLC1A3SLC1A2SLC1A1APP
SCHEMBL20889296 0.81 ALOX5 (0.59) ALOX5SLC1A3SLC1A2SLC1A1APP
SCHEMBL20509484 0.77 CYP1A2 (0.41) ALOX5SLC9A1SYKGPR139ADRA2A
SCHEMBL29985513 0.77 CYP1A2 (0.41) ALOX5SLC9A1SYKGPR139ADRA2A
SCHEMBL7366366 0.75 SLC1A3 (0.48) ALOX5SLC1A3SLC1A2SLC1A1CYP2C9
SCHEMBL19682744 0.75 SLC1A3 (0.48) ALOX5SLC1A3SLC1A2SLC1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
EP-3466934-A1 SULFONAMIDE COMPOUND OR SALT THEREOF Taiho Pharmaceutical Co., Ltd. (JP) 2019-04-10 EP disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 ALOX5 3456/4885SLC1A3 3645/4885SLC1A2 4159/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 ALOX5 3456/4885SLC1A3 3645/4885SLC1A2 4159/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 ALOX5 3456/4885SLC1A3 3645/4885SLC1A2 4159/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B ALOX5 3558/4885SLC1A3 3275/4885SLC1A2 4106/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.