SCHEMBL19684080

SCHEMBL19684080

COC(=O)[C@@H](NC(=O)c1ccc(C#CC#Cc2ccc(N)cc2)cc1)C(C)(N)C(F)F

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ACACB O00763 1/20 0.37
P2RY6 Q15077 1/20 0.36
MLYCD O95822 1/20 0.36
ADRB2 P07550 2/20 0.36
ADRB1 P08588 2/20 0.36
ADRB3 P13945 2/20 0.36
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
CA2 P00918 1/20 0.34
ESRRG P62508 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15235757 1.00 NPC1 (0.37) NPC1RAB9AACACBP2RY6MLYCD
SCHEMBL15237903 0.89 LMNA (0.36) NPC1RAB9AACACBP2RY6MLYCD
SCHEMBL15235731 0.89 ADRB2 (0.38) NPC1RAB9AACACBADRB2ADRB1
SCHEMBL19684304 0.88 ACACB (0.42) ACACBADRB2ADRB1ADRB3MAPT
SCHEMBL15235769 0.88 ACACB (0.42) ACACBADRB2ADRB1ADRB3MAPT
SCHEMBL19684253 0.87
SCHEMBL15228059 0.87
SCHEMBL15235759 0.87
SCHEMBL15235784 0.87
SCHEMBL15235729 0.86 CA2 (0.39) NPC1RAB9AACACBADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170349544-A1 Ethynylbenzene Derivatives DUKE UNIVERSITY 2017-12-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170349544-A1 Ethynylbenzene Derivatives Q6ZSR9, EPX, ZYX NPC1 2783/4885RAB9A 331/4885ACACB 2488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.