SCHEMBL19723151

SCHEMBL19723151

CC(C)n1cncc(C(C)(C)C)c1=O

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TNKS O95271 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL783436 0.75 GABRA5 (0.33)
SCHEMBL19723177 0.75 ALDH1A1 (0.34) ALDH1A1TDP1
SCHEMBL2621558 0.73 KDM5A (0.37) ALDH1A1TDP1
SCHEMBL24267978 0.73 ALDH1A1 (0.33) ALDH1A1TDP1
SCHEMBL23029116 0.73
SCHEMBL20847874 0.72 ALDH1A1 (0.32) ALDH1A1TDP1
SCHEMBL15185671 0.72 BMPR1B (0.36) ALDH1A1TDP1
SCHEMBL19723235 0.68 PTGS2 (0.36) ALDH1A1TDP1
SCHEMBL23229049 0.66 GSK3A (0.32)
SCHEMBL13988839 0.66 ADORA2A (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560967-B1 Heterocyclic carboxylic acid amides as PDK1 inihibitors BOEHRINGER INGELHEIM INT (DE) 2017-12-20 EP disclosed