SCHEMBL1973250

SCHEMBL1973250

NCCc1c[nH]c2cc3c(cc12)OCO3

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 11/20 0.66
HTR1D P28221 9/20 0.66
HTR1A P08908 7/20 0.66
HTR2C P28335 6/20 0.66
HTR1B P28222 6/20 0.66
HTR7 P34969 4/20 0.66
HTR6 P50406 4/20 0.66
HTR2B P41595 3/20 0.66
HTR4 Q13639 3/20 0.66
HTR3E A5X5Y0 2/20 0.66
HTR3B O95264 2/20 0.66
HTR1E P28566 2/20 0.66
HTR1F P30939 2/20 0.66
HTR3A P46098 2/20 0.66
HTR5A P47898 2/20 0.66
HTR3D Q70Z44 2/20 0.66
HTR3C Q8WXA8 2/20 0.66
MAPT P10636 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
ALDH1A1 P00352 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31079780 1.00 HTR2A (0.66) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL10773237 0.89 HTR2A (0.61) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL32669398 0.83 HTR1A (0.66) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL25747785 0.80 HTR2C (0.60) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL10770864 0.80 HTR1A (0.61) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL10772090 0.80 HTR1A (0.61) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL27077936 0.80 HTR2A (0.65) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL30249043 0.80 HTR1D (1.00) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL20970981 0.80 HTR1D (1.00) HTR2AHTR1DHTR1AHTR2CHTR1B
SCHEMBL32669266 0.77 MPO (0.59) HTR2AHTR1DHTR1AHTR2CHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334643-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES Actelion Pharmaceuticals Ltd. (CH) 2011-06-22 EP claimed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO claimed
EP-2334643-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES Actelion Pharmaceuticals Ltd. (CH) 2011-06-22 EP disclosed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed