SCHEMBL19732928

SCHEMBL19732928

Cc1ccc(S(=O)(=O)C(NC(N)=O)c2ccc(C#N)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
LMNA P02545 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 1/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
CYP2A6 P11509 1/20 0.41
KDM1A O60341 1/20 0.40
PRSS1 P07477 1/20 0.40
ACR P10323 1/20 0.40
FPR1 P21462 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
HCRTR2 O43614 1/20 0.40
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19732946 0.89 LMNA (0.51) CA12CA1CA2CA9LMNA
SCHEMBL19732939 0.83 TP53 (0.47) CA12CA1CA2CA9LMNA
SCHEMBL19732918 0.82 LMNA (0.59) CA12CA1CA2CA9LMNA
SCHEMBL19732963 0.81 ALDH1A1 (0.51) LMNAALDH1A1KMT2APRSS1
SCHEMBL19732931 0.80 ACHE (0.46) CA12CA1CA2CA9LMNA
SCHEMBL19732917 0.80 POLB (0.45) RORCCA12CA1CA2CA9
SCHEMBL16093818 0.79 KMT2A (0.46) RORCCA12CA1CA2CA9
SCHEMBL15913194 0.79 EEF2K (0.46) CA12CA1CA2CA9KDM1A
SCHEMBL19752704 0.78 KDM4E (0.35) CA12CA1CA2CA9LMNA
SCHEMBL19732921 0.77 MEN1 (0.44) CA12CA1CA2CA9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3260446-A1 ENANTIOSELECTIVE SYNTHESIS OF DIHYDROPYRIMIDINONES AND HEXAHYDROPYRIMIDINONES Universitat de les Illes Balears (ES) 2017-12-27 EP disclosed
EP-3260446-A1 ENANTIOSELECTIVE SYNTHESIS OF DIHYDROPYRIMIDINONES AND HEXAHYDROPYRIMIDINONES Universitat de les Illes Balears (ES) 2017-12-27 EP disclosed