SCHEMBL19732952

SCHEMBL19732952

COc1cccc([C@H]2NC(=O)NC(C)=C2C(=O)O)c1

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.69
ALDH1A1 P00352 3/20 0.66
L3MBTL1 Q9Y468 2/20 0.60
KDM4E B2RXH2 1/20 0.57
TP53 P04637 1/20 0.57
USP2 O75604 1/20 0.56
PDE1C Q14123 1/20 0.55
GUSB P08236 1/20 0.55
KIF11 P52732 1/20 0.54
EGFR P00533 1/20 0.53
HTT P42858 1/20 0.52
GAA P10253 1/20 0.52
THRB P10828 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14413854 1.00 NPSR1 (0.69) NPSR1ALDH1A1L3MBTL1KDM4ETP53
SCHEMBL19752619 0.85 KIF11 (0.75) NPSR1ALDH1A1L3MBTL1TP53PDE1C
SCHEMBL3395610 0.85 KIF11 (0.75) NPSR1ALDH1A1L3MBTL1TP53PDE1C
SCHEMBL19732926 0.84 ALDH1A1 (0.80) ALDH1A1KDM4ETP53USP2EGFR
SCHEMBL14413835 0.84 ALDH1A1 (0.80) ALDH1A1KDM4ETP53USP2EGFR
SCHEMBL3398149 0.83 KIF11 (0.71) NPSR1ALDH1A1L3MBTL1USP2GUSB
SCHEMBL19732923 0.82 USP2 (0.79) ALDH1A1KDM4ETP53USP2
SCHEMBL13789190 0.82 USP2 (0.79) ALDH1A1KDM4ETP53USP2
SCHEMBL19732955 0.82 USP2 (0.79) ALDH1A1KDM4ETP53USP2
SCHEMBL14413255 0.82 PKM (0.68) NPSR1ALDH1A1USP2GUSBKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3260446-A1 ENANTIOSELECTIVE SYNTHESIS OF DIHYDROPYRIMIDINONES AND HEXAHYDROPYRIMIDINONES Universitat de les Illes Balears (ES) 2017-12-27 EP disclosed