SCHEMBL19734693

SCHEMBL19734693

OC(c1cc(F)cc(F)c1)C1CN(CCC(F)F)C1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.38
CCL5 P13501 3/20 0.38
HTR2A P28223 5/20 0.37
HTR2C P28335 2/20 0.37
HTR7 P34969 2/20 0.37
CYP2D6 P10635 1/20 0.33
HTR6 P50406 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19734729 0.88 CCR5 (0.36) CCR5CCL5HTR2AHTR2CHTR7
SCHEMBL19731725 0.83 HTR2A (0.37) CCR5CCL5HTR2AHTR2CHTR7
SCHEMBL19731754 0.83 HTR2A (0.37) CCR5CCL5HTR2AHTR2CHTR7
SCHEMBL28195957 0.78 HTR2A (0.34) HTR2AHTR2CHTR7CYP2D6CES2
SCHEMBL18249584 0.74 CES2 (0.40) CCR5CCL5HTR2AHTR2CHTR7
SCHEMBL15609148 0.72 CES2 (0.41) HTR2AHTR2CHTR7CYP2D6HTR6
SCHEMBL18249640 0.70 CCL5 (0.36) CCR5CCL5
SCHEMBL19734482 0.69 CCL5 (0.31) CCR5CCL5
SCHEMBL19731647 0.69 CCL5 (0.31) CCR5CCL5
Oxalic Acid SCHEMBL18249620 0.67 CCR5 (0.39) CCR5CCL5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216280-A1 TETRAHYDRO-PYRIDO[3,4-b]INDOLE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-12-21 WO disclosed