SCHEMBL19735063

SCHEMBL19735063

CNSc1ccc(C=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.58
CYP2A6 P11509 4/20 0.46
TYR P14679 1/20 0.41
CYP2A13 Q16696 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ALDH5A1 P51649 1/20 0.41
ABAT P80404 1/20 0.41
ALDH1A3 P47895 2/20 0.39
ALDH3A1 P30838 1/20 0.39
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.33
EGFR P00533 1/20 0.33
TRIM24 O15164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
STS P08842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25014454 0.77 ALDH1A1 (0.50) ALDH1A1TSHR
SCHEMBL23912277 0.77 DRD1 (0.44) ALDH1A1CYP2A6TRIM24TRIM33
SCHEMBL195687 0.73 ALDH1A1 (1.00) ALDH1A1CYP2A6TYRCYP2A13HSD17B10
SCHEMBL224829 0.72 ALDH1A1 (0.64) ALDH1A1CYP2A6TYRCYP2A13HSD17B10
SCHEMBL6853611 0.72 ALDH1A1 (0.64) ALDH1A1CYP2A6TYRCYP2A13HSD17B10
SCHEMBL31171 0.71 CYP2A6 (0.69) ALDH1A1CYP2A6TYRCYP2A13HSD17B10
SCHEMBL4956384 0.71 CYP2A6 (0.69) ALDH1A1CYP2A6TYRCYP2A13HSD17B10
SCHEMBL13271224 0.70 ACHE (0.44) ALDH1A1
SCHEMBL24140273 0.69 ALDH1A1 (0.50) ALDH1A1HSD17B10TSHR
SCHEMBL20904129 0.69 ALDH1A1 (0.58) ALDH1A1CYP2A6TYRCYP2A13HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216727-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed
WO-2017216726-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed