Tangeretin

Tangeretin

SCHEMBL19740

COc1ccc(-c2cc(=O)c3c(OC)c(OC)c(OC)c(OC)c3o2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 1.00
MEN1 O00255 4/20 1.00
KMT2A Q03164 4/20 1.00
ABCB1 P08183 3/20 1.00
CYP3A4 P08684 2/20 1.00
ABCG2 Q9UNQ0 2/20 1.00
PKM P14618 1/20 1.00
MAPK1 P28482 2/20 0.80
PPARG P37231 2/20 0.80
MAPT P10636 3/20 0.71
KDM4E B2RXH2 2/20 0.71
HPGD P15428 1/20 0.71
HSD17B10 Q99714 1/20 0.71
TUBB4A P04350 1/20 0.65
TUBB P07437 1/20 0.65
TUBA3C P0DPH7 1/20 0.65
TUBA1B P68363 1/20 0.65
TUBA4A P68366 1/20 0.65
TUBB4B P68371 1/20 0.65
TUBB3 Q13509 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tangeretin SCHEMBL29549538 1.00 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AABCB1CYP3A4
Tangeretin SCHEMBL23629519 1.00 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AABCB1CYP3A4
Tangeretin SCHEMBL28155119 0.93 ALDH1A1 (0.87) ALDH1A1MEN1KMT2AABCB1CYP3A4
Gardenin B SCHEMBL1764516 0.89 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AABCB1CYP3A4
SCHEMBL31237871 0.89 ALDH1A1 (0.81) ALDH1A1MEN1KMT2AABCB1CYP3A4
SCHEMBL31570912 0.88 ALDH1A1 (0.78) ALDH1A1MEN1KMT2AABCB1CYP3A4
SCHEMBL30051182 0.87 PPARG (0.85) ALDH1A1MEN1KMT2AABCB1CYP3A4
SCHEMBL2622796 0.87 PPARG (0.85) ALDH1A1MEN1KMT2AABCB1CYP3A4
SCHEMBL12199707 0.87 ALDH1A1 (0.76) ALDH1A1MEN1KMT2AABCB1CYP3A4
SCHEMBL29187274 0.87 ALDH1A1 (0.76) ALDH1A1MEN1KMT2AABCB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5697 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121721044-B Online yarn hairiness detection system and method for texturing machine based on machine vision XI'AN HUODE IMAGE TECHNOLOGY Co.,Ltd. (CN) 2026-05-26 CN claimed
WO-2026107510-A1 HOT-MELT ADHESIVE COMPOSITION AND METHOD OF APPLICATION BIOBOND ADHESIVES, INC. (US) 2026-05-21 WO claimed
CN-122052146-A Self-adaptive power distribution method and system of hybrid energy storage system 西安热工研究院有限公司 2026-05-15 CN claimed
US-20260130395-A1 Water Dispersible Botanical Compositions AQUILA BLACK LTD (AU) 2026-05-14 US claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
US-20260096569-A1 EDIBLE COATING WITH ANTIMICROBIAL PROPERTIES APEEL TECH INC (US) 2026-04-09 US claimed
EP-4720261-A1 NOVEL CULTURE CONDITIONS FOR CLONAL EXPANSION OF NEPHRON PROGENITOR CELLS, GENERATION OF NEPHRON ORGANOIDS, AND RAPID AND SCALABLE MODELING OF POLYCYSTIC KIDNEY DISEASE University of Southern California (US) 2026-04-08 EP claimed
EP-4717264-A1 TANGERETIN FOR USE IN THE TREATMENT OF INFLAMMATORY DISEASES Xiangnan University (CN) 2026-04-01 EP claimed
EP-3346842-B1 STABLE INOCULANT COMPOSITIONS AND METHODS FOR PRODUCING SAME NOVONESIS PLANT BIOSOLUTIONS AS (DK) 2026-03-25 EP claimed
EP-4698662-A2 REGULATABLE CONTROLLED EXPRESSION OF A TRANSGENE IN PRIMATES AskBio Inc. (US) 2026-02-25 EP claimed
EP-0680744-B1 Use of flavonoid for hair protection OREAL (FR) 1999-09-29 EP claimed
EP-0605261-B1 Use of a flavone derivative as taste modifier and a method of modifying taste SAN EI GEN FFI INC (JP) 1999-09-15 EP claimed
EP-0938851-A2 Beverage and process for preparing it Eckes-Granini GmbH & Co. Kommanditgesellschaft (DE) 1999-09-01 EP claimed
WO-1999015167-A2 USE OF CITRUS LIMONOIDS AND FLAVONOIDS AS WELL AS TOCOTRIENOLS FOR THE TREATMENT OF CANCER KGK SYNERGIZE INC. (CA) 1999-04-01 WO claimed
EP-0627909-B1 COSMETIC OR PHARMACEUTICAL COMPOSITION CONTAINING A COMBINATION OF A POLYPHENOL AND A GINKGO EXTRACT OREAL (FR) 1999-03-03 EP claimed
WO-1998047534-A1 STABILIZED MEDICAMENTS CONTAINING CYSTEINYL DERIVATIVES KLINGE PHARMA GMBH (DE) 1998-10-29 WO claimed
US-5792448-A PROTECTING TENSILE STENGTH AND ELASTICITY OF HAIR BY APPLYING A COSMETIC CONTAINING FLAVONOIDS SUCH AS FLAVANONES, FLAVONES, FLAVONOLS, DIHYDROFLAVONOLS, CATECHINS AND LEUCOANTHOCYANIDINS L'OREAL (FR) 1998-08-11 US claimed
US-5686082-A AN ANTIOXIDIZING SYSTEM L'OREAL (FR) 1997-11-11 US claimed
US-5580545-A ADDING FLAVONE DERIVATIVES TO FOODS, BEVERAGES OR TOILETRIES TO ENHANCE OR REDUCE FLAVORS SAN-EI GEN F.F.I., INC. (JP) 1996-12-03 US claimed
EP-0605261-A2 A taste modifier and a method of modifying taste SAN-EI GEN F.F.I., INC. (JP) 1994-07-06 EP claimed