SCHEMBL19782394

SCHEMBL19782394

CCC(C)OC(=O)c1sc(Nc2ncccn2)nc1-c1ccncn1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 13/20 0.38
NOX1 Q9Y5S8 2/20 0.35
CYP3A4 P08684 1/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19782390 0.90 DHODH (0.36) DHODHNOX1CYP3A4MAPTKDM4E
SCHEMBL19783106 0.86 DHODH (0.53) DHODHMAPTKDM4EMEN1CYP1A2
SCHEMBL19782395 0.85 CDC7 (0.40) DHODHMAPTKDM4E
SCHEMBL19782392 0.84 DHODH (0.40) DHODHMAPTKDM4EMEN1CYP1A2
SCHEMBL19782989 0.84 DHODH (0.43) DHODHMAPTKDM4EMEN1CYP1A2
SCHEMBL19783003 0.78 ADORA3 (0.41) DHODHMAPTKDM4EMEN1CYP1A2
SCHEMBL19782384 0.74 ALDH1A1 (0.38) DHODHMAPTKDM4EMEN1CYP1A2
SCHEMBL15993345 0.74 DHODH (0.58) DHODHMAPTMEN1CYP1A2CYP2C9
SCHEMBL19782389 0.73 DHODH (0.38) DHODHMAPTKDM4EMEN1CYP1A2
SCHEMBL15993076 0.73 NPC1 (0.48) DHODHMAPTKDM4EKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013508-A1 SUBSTITUTED AMINOTHIAZOLES BARUCH S. BLUMBERG INSTITUTE (US) 2018-01-18 WO disclosed