SCHEMBL19783020

SCHEMBL19783020

O=CCCc1sc(NCc2ncccn2)nc1-c1ccccn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 2/20 0.36
ADAMTS4 O75173 1/20 0.36
MMP14 P50281 1/20 0.36
ADAMTS13 Q76LX8 1/20 0.36
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
NPC1 O15118 8/20 0.34
RAB9A P51151 7/20 0.34
MAPT P10636 7/20 0.34
KDM4E B2RXH2 6/20 0.34
SMN1; SMN2 Q16637 5/20 0.34
LMNA P02545 2/20 0.34
GAA P10253 2/20 0.34
HTT P42858 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
TP53 P04637 2/20 0.34
ALDH1A1 P00352 5/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ATM Q13315 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19783018 0.83 ADAMTS5 (0.50) ADAMTS5ADAMTS4MMP14ADAMTS13ADORA2A
SCHEMBL19783019 0.78 ALDH1A1 (0.42) ADAMTS5ADAMTS4MMP14ADAMTS13NPC1
SCHEMBL19782715 0.77 ADORA2A (0.40) ADORA2AADORA1NPC1RAB9AMAPT
SCHEMBL19783107 0.75 ALDH1A1 (0.47) NPC1RAB9AMAPTKDM4ESMN1; SMN2
SCHEMBL19782726 0.70 LMNA (0.56) ADORA2AADORA1NPC1RAB9AMAPT
SCHEMBL23965805 0.67 NPC1 (0.60) ADORA1NPC1RAB9AMAPTKDM4E
SCHEMBL19782991 0.66 MAPT (0.60) NPC1RAB9AMAPTKDM4ESMN1; SMN2
SCHEMBL27973907 0.66 KDR (0.36) ADAMTS5ADAMTS4MMP14ADAMTS13ADORA2A
SCHEMBL19782984 0.66 ADAMTS5 (0.52) ADAMTS5ADAMTS4MMP14ADAMTS13ADORA2A
SCHEMBL1017978 0.65 KMT2A (0.51) NPC1RAB9AMAPTKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013508-A1 SUBSTITUTED AMINOTHIAZOLES BARUCH S. BLUMBERG INSTITUTE (US) 2018-01-18 WO disclosed