SCHEMBL19783113

SCHEMBL19783113

Nc1nc(-c2ccccn2)c(CCO)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 8/20 0.49
PIK3CD O00329 1/20 0.43
PIK3CA P42336 1/20 0.43
PI4KA P42356 1/20 0.43
PIK3CG P48736 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
CYP1A2 P05177 1/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
RAB9A P51151 1/20 0.40
ALOX15 P16050 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
FBP1 P09467 1/20 0.39
ADAMTS4 O75173 1/20 0.39
MMP14 P50281 1/20 0.39
ADAMTS13 Q76LX8 1/20 0.39
ADAMTS5 Q9UNA0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18230383 0.85 ALDH1A1 (0.55) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL31361560 0.82 MAPT (0.62) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL2590963 0.78 ALDH1A1 (0.66) CYP1A2MAPTALDH1A1KDM4EL3MBTL1
SCHEMBL24358097 0.76 TGFBR1 (0.41) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL31361561 0.73 TGFBR1 (0.55) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL11796387 0.73 TGFBR1 (0.56) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL3737029 0.73 TGFBR1 (0.55) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
Bromide SCHEMBL29078717 0.72 TGFBR1 (0.54) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL5669674 0.72 TGFBR1 (0.50) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL1850971 0.70 TGFBR1 (0.51) TGFBR1PIK3CDPIK3CAPI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013508-A1 SUBSTITUTED AMINOTHIAZOLES BARUCH S. BLUMBERG INSTITUTE (US) 2018-01-18 WO disclosed