SCHEMBL19783296

SCHEMBL19783296

CN1C(O)N(Cc2ccccc2)C(=O)N1c1ccc2nn(-c3cccnc3)cc2c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 4/20 0.38
HPGD P15428 3/20 0.38
ESR2 Q92731 1/20 0.37
TLR8 Q9NR97 1/20 0.35
CACNA2D1 P54289 1/20 0.35
TP53 P04637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SNRNP200 O75643 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22172057 0.90 ALDH1A1 (0.34) ALDH1A1KDM4EHPGDTLR8L3MBTL1
SCHEMBL19783288 0.86 TLR8 (0.35) ESR2TLR8ADORA3
SCHEMBL21422303 0.85 TLR8 (0.39) ALDH1A1HPGDESR2TLR8CACNA2D1
SCHEMBL21422279 0.77 ALDH1A1 (0.39) ALDH1A1KDM4EESR2TLR8L3MBTL1
SCHEMBL19783974 0.72 POLB (0.38) ALDH1A1KDM4EESR2TLR8TP53
SCHEMBL19783856 0.72 ESR2 (0.41) ALDH1A1KDM4EESR2TLR8ADORA3
SCHEMBL19784122 0.71 GRIN1 (0.39) ALDH1A1KDM4EHPGDTLR8TP53
SCHEMBL19783865 0.71 TLR8 (0.39) ALDH1A1HPGDTLR8CACNA2D1HDAC1
SCHEMBL19784119 0.70 USP2 (0.39) ALDH1A1TLR8MEN1KMT2A
SCHEMBL19784121 0.70 HIF1A (0.39) ALDH1A1TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484877-B1 BICYCLIC COMPOUNDS AS PEST CONTROLLERS BAYER CROPSCIENCE AG (DE) 2020-07-01 EP disclosed
WO-2018011111-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-01-18 WO disclosed