SCHEMBL19787514

SCHEMBL19787514

NC1[C@@H]2C[C@H]1CN(c1ccnnc1)C2

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.38
CHRNA4 P43681 7/20 0.38
CHRNA7 P36544 2/20 0.38
CHRNB4 P30926 7/20 0.36
CHRNA3 P32297 7/20 0.36
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
MAPK3 P27361 1/20 0.33
MAPK1 P28482 1/20 0.33
PTPN11 Q06124 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21093913 0.91 CHRNB2 (0.37) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL21050385 0.90 CHRNB2 (0.40) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL21050383 0.90 CHRNB2 (0.40) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL21050384 0.90 CHRNB2 (0.40) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL23504818 0.75 CHRNA3 (0.36) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL16685011 0.73 HRH3 (0.44)
SCHEMBL23497916 0.72 PBK (0.45)
Hydrochloric Acid SCHEMBL16684779 0.71 HRH3 (0.42)
SCHEMBL20159697 0.71 APP (0.38) CHRNB2CHRNA4CHRNB4CHRNA3PSEN1
SCHEMBL20159656 0.71 CHRNA3 (0.39) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018011164-A1 FUSED PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2018-01-18 WO disclosed