SCHEMBL20159656

SCHEMBL20159656

N[C@@H]1[C@@H]2C[C@H]1CN(c1ccnc(Cl)c1)C2

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNA3 P32297 4/20 0.39
CHRNB2 P17787 4/20 0.39
CHRNB4 P30926 3/20 0.39
CHRNA4 P43681 3/20 0.39
CHRM4 P08173 1/20 0.39
MAPK3 P27361 1/20 0.38
MAPK1 P28482 1/20 0.38
PTPN11 Q06124 1/20 0.38
CHRM1 P11229 1/20 0.38
LOX P28300 1/20 0.36
LOXL3 P58215 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
CYP17A1 P05093 2/20 0.36
CHRNA7 P36544 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18970901 0.92 CHRM4 (0.38) CHRNA3CHRNB2CHRNB4CHRNA4CHRM4
SCHEMBL20609194 0.92 CHRM4 (0.38) CHRNA3CHRNB2CHRNB4CHRNA4CHRM4
SCHEMBL20609193 0.92 CHRM4 (0.38) CHRNA3CHRNB2CHRNB4CHRNA4CHRM4
SCHEMBL18952559 0.92 CHRM4 (0.38) CHRNA3CHRNB2CHRNB4CHRNA4CHRM4
SCHEMBL20031740 0.92 CHRM4 (0.38) CHRNA3CHRNB2CHRNB4CHRNA4CHRM4
SCHEMBL18971107 0.86 CHRNB4 (0.38) CHRNA3CHRNB2CHRNB4CHRNA4CHRM4
SCHEMBL20159647 0.78 CHRNB2 (0.40) CHRNA3CHRNB2CHRNB4CHRNA4CHRM1
SCHEMBL31614752 0.78 CHRM4 (0.41) CHRNA3CHRNB4CHRM4CHRM1LOX
SCHEMBL23504818 0.77 CHRNA3 (0.36) CHRNA3CHRNB2CHRNB4CHRNA4CHRNA7
SCHEMBL19787604 0.77 CHRM4 (0.43) CHRM4CHRM1LOXLOXL2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed