SCHEMBL19788967

SCHEMBL19788967

CCOC(=O)c1nn(C(C)(C)C)c2c1C1C(C)C(C)C1C2(F)F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
HPGD P15428 2/20 0.32
ELANE P08246 2/20 0.32
KDM4E B2RXH2 2/20 0.31
LMNA P02545 2/20 0.31
ALDH1A1 P00352 3/20 0.31
RAB9A P51151 2/20 0.31
NPC1 O15118 1/20 0.31
KMT2A Q03164 1/20 0.31
F2 P00734 1/20 0.31
PLAU P00749 1/20 0.31
MAPT P10636 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP1A2 P05177 1/20 0.31
TP53 P04637 1/20 0.30
ALOX12 P18054 1/20 0.30
CACNA1F O60840 1/20 0.30
CACNA1D Q01668 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20078937 0.82 LMNA (0.33) ADORA3ADORA2AADORA1ELANEKDM4E
SCHEMBL24878752 0.78 ALDH1A1 (0.35) HPGDELANEKDM4ELMNAALDH1A1
SCHEMBL19788768 0.78 KMT2A (0.32) ADORA3ADORA2AADORA1ELANEKDM4E
SCHEMBL17616500 0.78 KMT2A (0.32) ADORA3ADORA2AADORA1ELANEKDM4E
SCHEMBL17697354 0.66 PDE4A (0.36) ELANEKDM4ELMNAALDH1A1RAB9A
SCHEMBL21420081 0.66 MAPK1 (0.35) HPGDKDM4EALDH1A1KMT2AHSD17B10
SCHEMBL21420082 0.66 MAPK1 (0.35) HPGDKDM4EALDH1A1KMT2AHSD17B10
SCHEMBL4038348 0.66 ADORA3 (0.46) ADORA3ADORA2AADORA1HPGDELANE
SCHEMBL24998978 0.64 SMN1; SMN2 (0.30)
SCHEMBL22001985 0.64 MAPK1 (0.35) KDM4EALDH1A1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9873680-B2 Therapeutic compounds GILEAD SCIENCES, INC. (US) 2018-01-23 US disclosed