SCHEMBL19789660

SCHEMBL19789660

CC(=O)OC[C@@H]1C[C@H](OCc2ccccc2)[C@@H](OC(C)=O)[C@H](N=C=O)O1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
TSHR P16473 3/20 0.40
ALDH1A1 P00352 5/20 0.39
CYP2D6 P10635 3/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.37
CYP2C9 P11712 3/20 0.36
CYP3A4 P08684 3/20 0.36
MAPT P10636 2/20 0.36
CYP2C19 P33261 1/20 0.35
METAP2 P50579 2/20 0.35
BCHE P06276 1/20 0.34
GALR3 O60755 1/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976426 0.83 TSHR (0.45) LMNATSHRALDH1A1CYP2D6MAPK1
SCHEMBL13044308 0.83 TSHR (0.44) LMNATSHRALDH1A1CYP2D6MAPK1
SCHEMBL13044610 0.83 TSHR (0.44) LMNATSHRALDH1A1CYP2D6MAPK1
SCHEMBL13619819 0.80 CA12 (0.35) ALDH1A1CYP2D6CYP3A4MAPTCYP2C19
SCHEMBL404326 0.76 LMNA (0.42) LMNATSHRALDH1A1CYP2D6MAPK1
SCHEMBL19976411 0.75 BCHE (0.46) LMNATSHRALDH1A1BCHE
SCHEMBL14362881 0.74 LMNA (0.40) LMNATSHRALDH1A1CYP2D6MAPK1
SCHEMBL9522969 0.73 TSHR (0.51) LMNATSHRALDH1A1CYP2D6MAPK1
SCHEMBL10429257 0.73 TSHR (0.51) LMNATSHRALDH1A1CYP2D6MAPK1
SCHEMBL402667 0.73 ALDH1A1 (0.39) TSHRALDH1A1CYP3A4MAPTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282991-B1 METHOD FOR THE PRODUCTION OF 1,4-BENZOTHIEPIN-1,1-DIOXIDE DERIVATIVES SANOFI AVENTIS DEUTSCHLAND (DE) 2018-01-24 EP disclosed