SCHEMBL19790147

SCHEMBL19790147

CNC(Cc1c(F)c(F)c(F)c(F)c1F)C(C)=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.38
MMP2 P08253 2/20 0.37
MMP3 P08254 2/20 0.37
MMP1 P03956 1/20 0.37
OPRD1 P41143 1/20 0.34
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CTSL P07711 1/20 0.30
TAS1R3 Q7RTX0 1/20 0.30
TAS1R1 Q7RTX1 1/20 0.30
TAS1R2 Q8TE23 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14898392 1.00 CTSS (0.38) CTSSMMP2MMP3MMP1OPRD1
SCHEMBL25908942 0.93 TAS1R3 (0.37) CTSSMMP2MMP3MMP1OPRD1
SCHEMBL10065865 0.84 CTSS (0.41) CTSSMMP2MMP3MMP1OPRD1
SCHEMBL14949074 0.81 CTSS (0.37) CTSSMMP2MMP3MMP1OPRD1
SCHEMBL20364905 0.75 HDAC3 (0.38)
SCHEMBL19369908 0.74 MAOB (0.39)
SCHEMBL22679571 0.74 CTSS (0.33) CTSSMMP2MMP3MMP1PKM
SCHEMBL14898390 0.74 MAOB (0.39)
SCHEMBL18647237 0.73 ALDH1A1 (0.32) CTSSMMP2MMP3MMP1PKM
SCHEMBL26809260 0.73 ALDH1A1 (0.32) CTSSMMP2MMP3MMP1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937262-B1 COMPOSITION FOR USE IN TREATING GASTROINTESTINAL DYSMOTILITY IPSEN PHARMA (FR) 2019-05-08 EP disclosed
EP-2794634-B1 PROCESS FOR THE SYNTHESIS OF GHRELIN ANALOGUES IPSEN MFG IRELAND LIMITED (IE) 2018-01-24 EP disclosed