SCHEMBL19791848

SCHEMBL19791848

NS(=O)(=O)n1ccc2ncccc21

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MET P08581 13/20 0.64
RAPGEF4 Q8WZA2 1/20 0.56
RPS6KA5 O75582 3/20 0.49
CDC7 O00311 1/20 0.43
CDK2 P24941 1/20 0.43
RPS6KA4 O75676 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17194137 0.82 MET (0.64) METRAPGEF4RPS6KA5
SCHEMBL31428856 0.82 MET (0.64) METRAPGEF4RPS6KA5
SCHEMBL29847431 0.78 MET (1.00) METRAPGEF4
SCHEMBL3705420 0.78 MET (1.00) METRAPGEF4
SCHEMBL31405708 0.74 MET (0.62) METRAPGEF4RPS6KA5
SCHEMBL30711140 0.74 MET (0.76) METRAPGEF4
SCHEMBL3616325 0.74 MET (0.76) METRAPGEF4
SCHEMBL830432 0.74 ALDH3A1 (0.57)
SCHEMBL15175252 0.72 RAPGEF4 (1.00) METRAPGEF4
SCHEMBL16824192 0.71 MET (0.84) METRAPGEF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018015445-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY NodThera Limited (GB) 2018-01-25 WO disclosed
EP-3272739-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY NodThera Limited (GB) 2018-01-24 EP disclosed
EP-3272739-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY NodThera Limited (GB) 2018-01-24 EP disclosed