SCHEMBL1979322

SCHEMBL1979322

COc1ccc([N+](=O)[O-])c(-c2cc(Cl)ncc2Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MERTK Q12866 1/20 0.47
PIN1 Q13526 1/20 0.44
MAPT P10636 5/20 0.43
ALDH1A1 P00352 4/20 0.43
LMNA P02545 2/20 0.43
HPGD P15428 2/20 0.43
GFER P55789 2/20 0.43
MAPK1 P28482 2/20 0.43
RAF1 P04049 1/20 0.43
PAX8 Q06710 1/20 0.43
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
S1PR4 O95977 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1984450 0.87 MERTK (0.38) MERTKPIN1MAPTALDH1A1LMNA
SCHEMBL1984451 0.87 MAPT (0.41) MERTKMAPTALDH1A1LMNAHPGD
SCHEMBL11199415 0.81 ALDH1A1 (0.54) MERTKMAPTALDH1A1LMNAHPGD
SCHEMBL12597604 0.81 FFAR4 (0.37) MERTKPIN1MAPK1KMT2ANPC1
SCHEMBL1983238 0.76 HSP90AA1 (0.47) MAPTALDH1A1HPGDGFERMAPK1
SCHEMBL1629413 0.75 MAPK1 (0.58) MERTKPIN1MAPTALDH1A1LMNA
SCHEMBL30310607 0.75 MAPK1 (0.58) MERTKPIN1MAPTALDH1A1LMNA
SCHEMBL1979039 0.74 ALDH1A1 (0.47) PIN1MAPTALDH1A1LMNAHPGD
SCHEMBL22604633 0.73 MERTK (0.56) MERTKPIN1MAPTALDH1A1LMNA
SCHEMBL541479 0.72 ALDH1A1 (0.68) MERTKMAPTALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed