SCHEMBL1979335

SCHEMBL1979335

COC(C)Oc1cccc([N+](=O)[O-])c1-c1cc(Cl)ncc1Cl

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 5/20 0.37
ALDH1A1 P00352 4/20 0.36
TDP1 Q9NUW8 3/20 0.36
HPGD P15428 1/20 0.36
NR1H4 Q96RI1 1/20 0.35
EGFR P00533 1/20 0.34
S100A4 P26447 2/20 0.34
PTPRC P08575 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
HSD11B1 P28845 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
MAPK1 P28482 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979039 0.87 ALDH1A1 (0.47) PIN1ALDH1A1TDP1HPGDEGFR
SCHEMBL1979336 0.82 NPC1 (0.44) PIN1ALDH1A1HPGDEGFRKDM4E
SCHEMBL1984450 0.77 MERTK (0.38) PIN1ALDH1A1TDP1HPGDMEN1
SCHEMBL1978964 0.77 SCD (0.39) PIN1ALDH1A1TDP1HPGDEGFR
SCHEMBL10583683 0.70 ALDH1A1 (0.65) ALDH1A1TDP1HPGDMEN1KMT2A
SCHEMBL1979322 0.68 MERTK (0.47) PIN1ALDH1A1TDP1HPGDKDM4E
SCHEMBL10582382 0.67 ALDH1A1 (0.59) ALDH1A1TDP1HPGDMEN1KMT2A
SCHEMBL15283821 0.66 PDK1 (0.45) PIN1TDP1EGFRMEN1KMT2A
SCHEMBL27952716 0.64 ALDH1A1 (0.63) ALDH1A1TDP1HPGDKDM4EMEN1
SCHEMBL30991376 0.64 ALDH1A1 (0.58) PIN1ALDH1A1TDP1HPGDS100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed