SCHEMBL19794945

SCHEMBL19794945

Nc1cc2cc(F)ccc2o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA9 Q16790 1/20 0.50
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
APP P05067 1/20 0.41
PLAU P00749 1/20 0.40
BACE1 P56817 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2A6 P11509 1/20 0.38
PGR P06401 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
FLT3 P36888 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3920685 0.77 FLT3 (0.59) CA2CHRM2CHRM4CHRM5CHRM1
SCHEMBL14231750 0.77 CHRM2 (0.54) CA2CA12CA1CA9CHRM2
SCHEMBL11831412 0.76 CA12 (0.61) CA2CA12CA1CA9PLAU
SCHEMBL8037247 0.74 CDK9 (0.50) CA2CA12CA1CA9CHRM2
SCHEMBL18233454 0.74 CA12 (0.46) CA2CA12CA1CA9CHRM2
SCHEMBL18003606 0.74 CA12 (0.46) CA2CA12CA1CA9CHRM2
SCHEMBL12267 0.74 DYRK1A (0.50) CA2CA12CA1CA9CHRM2
SCHEMBL12347 0.74 ALDH1A1 (0.52) CA2CA12CA1CA9ALDH1A1
SCHEMBL15031527 0.74 MAOB (0.55) CA2CA12CA1CA9APP
SCHEMBL20210894 0.74 CA12 (0.46) CA2CA12CA1CA9CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022079092-A1 TETRAZOLE DERIVATIVES AS TRPA1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-04-21 WO disclosed
WO-2022079091-A1 TETRAZOLE DERIVATIVES AS TRPA1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-04-21 WO disclosed
WO-2018015410-A1 BICYCLIC PROLINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2018-01-25 WO disclosed