SCHEMBL1979799

SCHEMBL1979799

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(C(=O)NCC(C)N2CCCC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.41
MAPT P10636 2/20 0.41
CHEK1 O14757 1/20 0.40
ACHE P22303 1/20 0.40
LMNA P02545 4/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
NEK1 Q96PY6 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
TLR7 Q9NYK1 1/20 0.38
DYRK1A Q13627 1/20 0.38
SMPD1 P17405 1/20 0.38
PIM1 P11309 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979088 0.87 WNT1 (0.51) CHEK1ACHETLR7DYRK1A
SCHEMBL1981901 0.86 CHEK1 (0.40) CHEK1ACHEROCK2ROCK1ALDH1A1
SCHEMBL12598125 0.86 DRD2 (0.48) MAPTSMN1; SMN2CYP1A2CYP2C19TLR7
SCHEMBL473769 0.85 CHEK1 (0.45) TP53MAPTCHEK1ACHELMNA
SCHEMBL1983761 0.85 BRAF (0.47) TP53MAPTALDH1A1TLR7DYRK1A
SCHEMBL1981803 0.84 MTNR1A (0.45) ALDH1A1CYP1A2TLR7SMPD1PIM1
SCHEMBL12597223 0.84 TLR7 (0.42) ALDH1A1TLR7DYRK1ASMPD1PIM1
SCHEMBL12597359 0.84 SLC2A1 (0.45) NEK1TLR7SMPD1PIM1
SCHEMBL1981315 0.83 PTAFR (0.47) TP53ALDH1A1TLR7DYRK1ASMPD1
SCHEMBL12598121 0.83 KDM4E (0.44) TP53MAPTALDH1A1TLR7DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed