SCHEMBL1979088

SCHEMBL1979088

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(C(=O)NCCN2CCCCCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
WNT1 P04628 3/20 0.51
DYRK1A Q13627 3/20 0.51
TLR9 Q9NR96 3/20 0.49
TLR7 Q9NYK1 3/20 0.49
TLR8 Q9NR97 2/20 0.48
CHEK1 O14757 1/20 0.47
ACHE P22303 1/20 0.47
PARP1 P09874 1/20 0.46
HTR3A P46098 1/20 0.45
ABL1 P00519 2/20 0.43
BCR P11274 2/20 0.43
IGF1R P08069 1/20 0.42
F10 P00742 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA1A P35348 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12598125 0.94 DRD2 (0.48) WNT1DYRK1ATLR9TLR7TLR8
SCHEMBL12598121 0.89 KDM4E (0.44) WNT1DYRK1ATLR9TLR7TLR8
SCHEMBL1983761 0.88 BRAF (0.47) WNT1DYRK1ATLR9TLR7
SCHEMBL1980365 0.87 TLR7 (0.52) WNT1DYRK1ATLR9TLR7TLR8
SCHEMBL1981803 0.87 MTNR1A (0.45) TLR9TLR7TLR8
SCHEMBL1979799 0.87 TP53 (0.41) DYRK1ATLR7CHEK1ACHE
SCHEMBL1979171 0.86 WNT1 (0.42) WNT1DYRK1ATLR9TLR7TLR8
SCHEMBL1981315 0.86 PTAFR (0.47) WNT1DYRK1ATLR9TLR7
SCHEMBL1981901 0.86 CHEK1 (0.40) WNT1DYRK1ATLR9TLR7TLR8
SCHEMBL12598112 0.86 TLR7 (0.45) DYRK1ATLR9TLR7TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed