SCHEMBL19798045

SCHEMBL19798045

N#Cc1ccc(-c2ccc(CC(=O)Cc3ccc(-c4ccc(F)cc4)cc3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 2/20 0.51
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
CTBP2 P56545 1/20 0.47
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
VNN1 O95497 1/20 0.46
RXRA P19793 1/20 0.46
RXRG P48443 1/20 0.46
MMP12 P39900 1/20 0.46
MMP13 P45452 1/20 0.46
MMP3 P08254 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
PTGDR2 Q9Y5Y4 2/20 0.43
MMP2 P08253 1/20 0.43
PTGS1 P23219 1/20 0.43
EPHX2 P34913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9190571 0.95 NSD2 (0.55) NSD2MAOAMAOBCTBP2CYP11B1
SCHEMBL6937899 0.86 CTBP2 (0.59) CTBP2MMP12MMP13SAE1UBA2
SCHEMBL27675295 0.86 GAA (0.52) MAOBCTBP2RXRARXRGKDM4E
SCHEMBL17857804 0.82 KMT2A (0.58) NSD2MAOAMAOBCTBP2CYP11B1
SCHEMBL526194 0.80 GAA (0.57) CTBP2KDM4EALDH1A1POLBGAA
SCHEMBL7929151 0.80 MMP3 (0.58) MAOAMAOBCYP11B1CYP11B2MMP3
SCHEMBL20941548 0.79 GAA (0.60) POLBGAASAE1UBA2TSHR
SCHEMBL8185095 0.79 HTT (0.62) CTBP2RXRARXRGMMP12MMP13
SCHEMBL9641208 0.79 CTBP2 (0.57) MAOAMAOBCTBP2SAE1UBA2
SCHEMBL17857729 0.77 TSHR (0.62) NSD2MAOAMAOBCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180022996-A1 BIMESOGENIC COMPOUNDS AND MESOGENIC MEDIA MERCK PATENT GMBH (DE) 2018-01-25 US disclosed
US-20180022996-A1 BIMESOGENIC COMPOUNDS AND MESOGENIC MEDIA MERCK PATENT GMBH (DE) 2018-01-25 US disclosed