SCHEMBL1980545

SCHEMBL1980545

Brc1ccc(-c2[c]cccn2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 2/20 0.38
RAB9A P51151 5/20 0.37
NPC1 O15118 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
KDM4E B2RXH2 2/20 0.37
TP53 P04637 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
HTT P42858 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
MEN1 O00255 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1202054 0.81 NOTUM (0.37) ALDH1A1MAPK1RAB9ANPC1SMN1; SMN2
SCHEMBL1973038 0.80 MAPK14 (0.36) ALDH1A1RAB9ANPC1MAPTHPGD
SCHEMBL5539865 0.80 NISCH (0.37) ALDH1A1RAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL435455 0.80 CYP1A2 (0.38) ALDH1A1MAPK1RAB9ANPC1SMN1; SMN2
SCHEMBL2397171 0.79 MAPT (0.42) ALDH1A1RAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL5544984 0.76 KIF11 (0.47) NPC1MAPTCCNB2CDK1CCNB1
SCHEMBL11240403 0.76 MAPT (0.46) ALDH1A1MAPK1RAB9ANPC1SMN1; SMN2
SCHEMBL5290073 0.76 CYP11B2 (0.43) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL5541420 0.76 CYP17A1 (0.41) ALDH1A1MAPK1RAB9ANPC1KDM4E
SCHEMBL1967426 0.76 CLK4 (0.56) ALDH1A1RAB9ANPC1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072207-A1 AZOCYCLIC INHIBITORS OF FATTY ACID AMIDE HYDROLASE E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-06-16 WO disclosed
EP-1909775-A2 FORMULATION OF RADIOPROTECTIVE ALPHA, BETA UNSATURATED ARYL SULFONES Onconova Therapeutics, Inc. (US) 2008-04-16 EP disclosed
WO-2007016201-A2 FORMULATION OF RADIOPROTECTIVE α, β UNSATURATED ARYL SULFONES ONCONOVA THERAPEUTICS, INC. (US) 2007-02-08 WO disclosed