SCHEMBL1981985

SCHEMBL1981985

CN1C(=O)NC2(CC(C)(Cc3ccc(F)cc3)Oc3ccc(Br)cc32)C1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 13/20 0.40
CTSD P07339 2/20 0.40
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.33
ITGAL P20701 2/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
FPR2 P25090 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1982116 0.86 MAOB (0.32) BACE1CTSDITGALITGB2ICAM1
SCHEMBL1979002 0.84 AKR1B1 (0.45) MAPT
SCHEMBL1983002 0.83 BACE1 (0.40) BACE1CTSDALDH1A1HPGDTP53
SCHEMBL1982797 0.82 MEN1 (0.39) BACE1CTSD
SCHEMBL1985921 0.78 BACE1 (0.39) BACE1
SCHEMBL1983498 0.75 BACE1 (0.47) BACE1CTSDALDH1A1HPGDMAPT
SCHEMBL1982412 0.75 BACE1 (0.46) BACE1CTSDMAPT
SCHEMBL1978797 0.70 BACE1 (0.46) BACE1MAPT
SCHEMBL1978518 0.70 AKT1 (0.44) ALDH1A1HPGDMAPT
SCHEMBL1978781 0.70 AKR1B1 (0.40) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed