SCHEMBL1983002

SCHEMBL1983002

CN1C(=O)NC2(CC(C)(Cc3cccnc3)Oc3ccc(Br)cc32)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.40
CTSD P07339 2/20 0.40
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
RIPK1 Q13546 1/20 0.36
MEN1 O00255 1/20 0.36
PKM P14618 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
GABRA1 P14867 1/20 0.34
GABRA5 P31644 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1983498 0.92 BACE1 (0.47) BACE1CTSDCYP1A2CYP3A4CYP2D6
SCHEMBL1978029 0.85 CYP3A4 (0.37) BACE1CTSDCYP1A2CYP3A4CYP2D6
SCHEMBL1981985 0.83 BACE1 (0.40) BACE1CTSDALDH1A1HPGDTP53
SCHEMBL1982797 0.83 MEN1 (0.39) BACE1CTSDMEN1KMT2APOLB
SCHEMBL1982412 0.76 BACE1 (0.46) BACE1CTSDMEN1KMT2A
SCHEMBL1982116 0.73 MAOB (0.32) BACE1CTSD
SCHEMBL1978480 0.72 KDM4E (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL12592601 0.69 BACE1 (0.70) BACE1CTSD
SCHEMBL1978759 0.68 MEN1 (0.36) MEN1KMT2A
SCHEMBL1978797 0.68 BACE1 (0.46) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed