SCHEMBL19823041

SCHEMBL19823041

Cc1cccn2cc(C3CC3)nc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 12/20 0.55
NPC1 O15118 11/20 0.55
ALDH1A1 P00352 11/20 0.55
KDM4E B2RXH2 11/20 0.55
SMN1; SMN2 Q16637 6/20 0.55
HSD17B10 Q99714 5/20 0.55
HPGD P15428 4/20 0.55
TP53 P04637 2/20 0.55
NPSR1 Q6W5P4 2/20 0.55
TSHR P16473 1/20 0.55
NFKB1 P19838 3/20 0.54
NFKB2 Q00653 3/20 0.54
RELA Q04206 3/20 0.54
GAA P10253 2/20 0.54
PKM P14618 2/20 0.51
PDE10A Q9Y233 1/20 0.50
PDE8B O95263 1/20 0.46
MAPT P10636 4/20 0.45
MAPK1 P28482 2/20 0.45
POLB P06746 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7551994 0.93 RAB9A (0.49) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL7510832 0.90 ALDH1A1 (0.49) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL7505996 0.86 KDM4E (0.46) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL7506673 0.84 DRD2 (0.46) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL17237851 0.83 RAB9A (0.55) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL7508321 0.82 HRH3 (0.48) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL7507239 0.82 DRD2 (0.52) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL15766578 0.81 PDE10A (0.51) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL15767328 0.80 PDE10A (0.77) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL21695773 0.78 ALDH1A1 (0.47) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2919783-B1 CYCLOPROPYL IMIDAZOPYRIDINE PDE10 INHIBITORS MERCK SHARP & DOHME (US) 2018-01-31 EP disclosed