SCHEMBL7507239

SCHEMBL7507239

Cc1cccn2cc(C3CCN(Cc4ccccc4)CC3)nc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.52
DRD4 P21917 11/20 0.52
DRD3 P35462 11/20 0.52
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
TP53 P04637 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ACHE P22303 1/20 0.46
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7505996 0.85 KDM4E (0.46) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL7506673 0.83 DRD2 (0.46) DRD2ALDH1A1KDM4ENPC1RAB9A
SCHEMBL19823041 0.82 RAB9A (0.55) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL5077376 0.81 GAA (0.45) DRD2DRD4DRD3POLB
SCHEMBL7508321 0.81 HRH3 (0.48) DRD2DRD3ALDH1A1KDM4ENPC1
SCHEMBL7510832 0.81 ALDH1A1 (0.49) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL5252888 0.79 MEN1 (0.42) DRD2DRD4DRD3KDM4ENPC1
SCHEMBL7551994 0.76 RAB9A (0.49) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL13490557 0.75 DRD2 (0.59) DRD2DRD4DRD3ACHEMEN1
SCHEMBL13490648 0.73 DRD2 (0.60) DRD2DRD4DRD3ACHEMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257551-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-11-20 EP disclosed
WO-2001057038-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-08-09 WO disclosed