Benzthiazide

Benzthiazide

SCHEMBL198231

NC(CS)C(=O)O.NS(=O)(=O)c1cc2c(cc1Cl)N=C(CSCc1ccccc1)NS2(=O)=O

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC12A3

The experimentally established mechanism targets of Benzthiazide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 1/20 0.52
MEN1 O00255 1/20 0.52
NR1I2 O75469 1/20 0.52
ABCB11 O95342 1/20 0.52
CYP3A4 P08684 1/20 0.52
ADRA2A P08913 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
PKM P14618 1/20 0.52
TSHR P16473 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
KMT2A Q03164 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
CA1 P00915 14/20 0.39
CA2 P00918 14/20 0.39
CA12 O43570 12/20 0.39
CA9 Q16790 11/20 0.39
CA6 P23280 10/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzthiazide SCHEMBL2452168 0.90 ALDH1A1 (0.51) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL2449654 0.90 ALDH1A1 (0.51) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL26257 0.89 ALDH1A1 (0.63) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL936396 0.89 ALDH1A1 (0.49) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL1276519 0.89 ALDH1A1 (0.60) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL345215 0.89 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL7217920 0.89 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL9517821 0.89 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL7102453 0.89 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL6546528 0.89 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 419 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11965198-B2 Method for producing target substance by bacterial fermentation AJINOMOTO CO., INC. (JP) 2024-04-23 US disclosed
EP-4291182-A1 MICROBIAL ERGOTHIONEINE BIOSYNTHESIS Conagen Inc. (US) 2023-12-20 EP disclosed
US-20220010343-A1 Method of Producing L-Amino Acids AJINOMOTO CO., INC. (JP) 2022-01-13 US disclosed
US-11198894-B2 Method of producing an l-amino acid involving a carotenoid biosynthesis enzyme AJINOMOTO CO., INC. (JP) 2021-12-14 US disclosed
EP-3861109-A1 METHOD FOR PRODUCING TARGET SUBSTANCE BY BACTERIAL FERMENTATION AJINOMOTO CO., INC. (JP) 2021-08-11 EP disclosed
WO-2021060438-A1 METHOD FOR PRODUCING L-AMINO ACIDS BY BACTERIAL FERMENTATION AJINOMOTO CO., INC. (JP) 2021-04-01 WO disclosed
EP-3098319-B1 A METHOD FOR PRODUCING AN L-AMINO ACID USING A BACTERIUM OF THE FAMILY ENTEROBACTERIACEAE HAVING AN ATTENUATED EXPRESSION OF A GSHA GENE AJINOMOTO KK (JP) 2020-11-25 EP disclosed
WO-2020204179-A1 METHOD OF PRODUCING L-AMINO ACIDS AJINOMOTO CO., INC. (JP) 2020-10-08 WO disclosed
EP-3385389-B1 METHOD FOR PRODUCING L-AMINO ACIDS FROM FRUCTOSE AJINOMOTO KK (JP) 2020-10-07 EP disclosed
US-10787691-B2 Method for producing L-amino acid AJINOMOTO CO., INC. (JP) 2020-09-29 US disclosed
US-20030199088-A1 For the production of achromosomal archeabacterial, eubacterial and anucleate eukaryotic cells; for therapeutics, diagnostics, drug discovery, proteomics VAXIION THERAPEUTICS, LLC 2003-10-23 US disclosed
US-20030194714-A1 Minicell-based transformation MPEX BIOSCIENCES, INC. 2003-10-16 US disclosed
US-20030194798-A1 For diagnositic, therapeutic, research, and drug discovery applications MPEX BIOSCIENCES, INC. 2003-10-16 US disclosed
US-20030190749-A1 Expression element that comprises a gene linked to sequences that are inducible and/or repressible; mutations; useful in diagnositics, therapeutics and drug discovery MPEX BIOSCIENCES, INC. 2003-10-09 US disclosed
US-20030190601-A1 Useful for diagnosis and therapy, research tools for drug discovery MPEX BIOSCIENCES, INC. 2003-10-09 US disclosed
US-20030190683-A1 Production of achromosomal and anucleate cells useful for diagnositic and therapeutic uses, as well as research tools and agents for drug discovery MPEX BIOSCIENCES, INC. 2003-10-09 US disclosed
US-20030166099-A1 Minicells comprising membrane proteins MPEX BIOSCIENCES, INC. 2003-09-04 US disclosed
US-20030166279-A1 Cell culture incubation and transferring nucleic acid from a minicell to a cell; diagnositic and therapeutic uses, as research tools and agents for drug discovery screening MPEX BIOSCIENCES, INC. 2003-09-04 US disclosed
WO-2003072014-A2 MINICELL COMPOSITIONS AND METHODS MPEX BIOSCIENCE, INC. (US) 2003-09-04 WO disclosed
WO-2002094867-A2 SEQUENCE OF THE PHOTORHABDUS LUMINESCENS STRAIN TT01 GENOME AND USES INSTITUT PASTEUR (FR) 2002-11-28 WO disclosed