Benzthiazide

Benzthiazide

SCHEMBL936396

CSCC[C@H](N)C(=O)O.NS(=O)(=O)c1cc2c(cc1Cl)N=C(CSCc1ccccc1)NS2(=O)=O

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC12A3

The experimentally established mechanism targets of Benzthiazide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
NR1I2 O75469 1/20 0.49
ABCB11 O95342 1/20 0.49
CYP3A4 P08684 1/20 0.49
ADRA2A P08913 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
PKM P14618 1/20 0.49
TSHR P16473 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CA1 P00915 9/20 0.38
CA2 P00918 9/20 0.38
CA12 O43570 8/20 0.37
CA6 P23280 8/20 0.37
CA7 P43166 8/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzthiazide SCHEMBL2452168 0.89 ALDH1A1 (0.51) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL2449654 0.89 ALDH1A1 (0.51) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL198231 0.89 ALDH1A1 (0.52) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL26257 0.87 ALDH1A1 (0.63) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL2376967 0.86 ALDH1A1 (0.58) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL386199 0.86 ALDH1A1 (0.46) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL1276519 0.86 ALDH1A1 (0.60) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL7102453 0.86 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL345215 0.86 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11
Benzthiazide SCHEMBL7217920 0.86 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 154 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024008889-A1 RECOMBINANT HOST CELLS PRODUCING IRONES AND USES THEREOF MUSEUM NATIONAL D'HISTOIRE NATURELLE (FR) 2024-01-11 WO disclosed
EP-4303308-A1 RECOMBINANT HOST CELLS PRODUCING IRONES AND USES THEREOF MUSEUM NATIONAL D'HISTOIRE NATURELLE (FR) 2024-01-10 EP disclosed
US-11845964-B2 Bacteria engineered to treat diseases associated with hyperammonemia SYNLOGIC OPERATING COMPANY, INC. (US) 2023-12-19 US disclosed
US-11390896-B2 Method for producing L-methionine using a bacterium of the genus Pantoea AJINOMOTO CO., INC. (JP) 2022-07-19 US disclosed
EP-3940067-A1 BACTERIA ENGINEERED TO TREAT DISEASES ASSOCIATED WITH HYPERAMMONEMIA Synlogic Operating Company, Inc. (US) 2022-01-19 EP disclosed
EP-3856918-A1 METHOD FOR PRODUCING L-METHIONINE USING A BACTERIUM AJINOMOTO CO., INC. (JP) 2021-08-04 EP disclosed
EP-3227440-B1 BACTERIA ENGINEERED TO TREAT DISEASES ASSOCIATED WITH HYPERAMMONEMIA SYNLOGIC OPERATING CO INC (US) 2021-07-14 EP disclosed
US-11060073-B2 Bacteria engineered to treat diseases associated with hyperammonemia SYNLOGIC OPERATING COMPANY, INC. (US) 2021-07-13 US disclosed
US-20210207182-A1 METHOD FOR PRODUCING L-METHIONINE USING A BACTERIUM AJINOMOTO CO., INC. (JP) 2021-07-08 US disclosed
US-20210180033-A1 BACTERIA ENGINEERED TO TREAT DISEASES ASSOCIATED WITH HYPERAMMONEMIA SYNLOGIC OPERATING COMPANY, INC. 2021-06-17 US disclosed
EP-1526179-B1 Method for producing l-amino acid using bacteria belonging to the genus escherichia AJINOMOTO KK (JP) 2007-05-02 EP disclosed
EP-1747269-A2 RECOMBINANT ENZYME WITH ALTERED FEEDBACK SENSITIVITY Metabolic Explorer (FR) 2007-01-31 EP disclosed
WO-2006082254-A2 MICROORGANISMS COMPRISING ENZYMES EXPRESSED WITH LOW GAMMA-ELIMINATION ACTIVITY METABOLIC EXPLORER (FR) 2006-08-10 WO disclosed
WO-2006082252-A2 METHOD FOR THE ENZYMATIC PRODUCTION OF ALPHA-KETOBUTYRATE METABOLIC EXPLORER (FR) 2006-08-10 WO disclosed
EP-1239041-B1 Method for producing L-amino acid using bacteria belonging to the genus Escherichia AJINOMOTO KK (JP) 2006-04-19 EP disclosed
WO-2005108561-A2 RECOMBINANT ENZYME WITH ALTERED FEEDBACK SENSITIVITY METABOLIC EXPLORER (FR) 2005-11-17 WO disclosed
US-20050239175-A1 Method for producing L-amino acid using bacteria belonging to the genus Escherichia AJINOMOTO CO., INC. (JP) 2005-10-27 US disclosed
EP-1526179-A1 Method for producing l-amino acid using bacteria belonging to the genus escherichia Ajinomoto Co., Inc. (JP) 2005-04-27 EP disclosed
EP-1526181-A1 Method for producing l-amino acid using bacteria belonging to the genus escherichia Ajinomoto Co., Inc. (JP) 2005-04-27 EP disclosed
EP-1239041-A2 Method for producing L-amino acid using bacteria belonging to the genus Escherichia Ajinomoto Co., Inc. (JP) 2002-09-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11845964-B2 Bacteria engineered to treat diseases associated with hyperammonemia ASS1, AGXT, OAT ALDH1A1 1080/4885KDM4E 3926/4885MEN1 787/4885
US-11060073-B2 Bacteria engineered to treat diseases associated with hyperammonemia ASS1, AGXT, OAT ALDH1A1 1080/4885KDM4E 3926/4885MEN1 787/4885
US-20210180033-A1 BACTERIA ENGINEERED TO TREAT DISEASES ASSOCIATED WITH HYPERAMMONEMIA ASS1, AGXT, OAT ALDH1A1 1080/4885KDM4E 3926/4885MEN1 787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.